Preparation of quinazolino[3,2-a]quinazolines via a palladium-catalyzed three-component reaction of carbodiimide, isocyanide, and amine.

نویسندگان

  • Guanyinsheng Qiu
  • Yaohua He
  • Jie Wu
چکیده

A palladium-catalyzed three-component reaction of bis-(2-iodoaryl)carbodiimide, isocyanide, and amine gives rise to quinazolino[3,2-a]quinazolines and related compounds in good yields. Multi-bonds are formed in one pot through nucleophilic attack, isocyanide insertion, and C-N coupling during the reaction process.

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عنوان ژورنال:
  • Chemical communications

دوره 48 32  شماره 

صفحات  -

تاریخ انتشار 2012